TGase2-IN-1
TGase2-IN-1 (Compound 22) is an orally active inhibitor for TGase2 with an IC50 of 1.12 μM. TGase2-IN-1 inhibits TGase2 in human retinal microvascular endothelial cells with an IC50 of 0.07 μM. TGase2-IN-1 exhibits 74.6% oral bioavailability. TGase2-IN-1 inhibits retinal vascular leakage in mouse Streptozotocin (HY-13753)-induced diabetic model.
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- CAS No.: 2244702-64-3
- Formule: C23H25N3O3
- Masse moléculaire:391.46
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Stockage:
Please store the product under the recommended conditions in the Certificate of Analysis.
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Activité biologique
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Chemical Information
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Activité biologique
Chemical Information
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CAS No. 2244702-64-3
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Masse moléculaire 391.46
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Formule C23H25N3O3
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SMILES
O=C1C=C(C(C2=NC(C3=CC=C(OC4CCN(C(C)C)CC4)C=C3)=CC=C12)=O)N
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Livraison
Room temperature in continental US; may vary elsewhere.
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Stockage
Please store the product under the recommended conditions in the Certificate of Analysis.
Pureté et documentation
Références
Calculators
Concentration (start) × Volume (start) = Concentration (final) × Volume (final)
TGase2-IN-1 Related Classifications
HY-159962 Related Classifications
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