1. GPCR/G Protein
    Neuronal Signaling
  2. Adrenergic Receptor
    Dopamine Receptor

Piribedil 

Cat. No.: HY-12707 Purity: 99.90%
Handling Instructions

Piribedil is a dopamine D2 receptor (D2R) agonist which also displays antagonist property at 1A-adrenoceptor (1A-AR).

For research use only. We do not sell to patients.

Piribedil Chemical Structure

Piribedil Chemical Structure

CAS No. : 3605-01-4

Size Price Stock Quantity
Free Sample (0.5-1 mg)   Apply now  
10 mM * 1 mL in DMSO USD 66 In-stock
Estimated Time of Arrival: December 31
10 mg USD 60 In-stock
Estimated Time of Arrival: December 31
50 mg USD 90 In-stock
Estimated Time of Arrival: December 31
100 mg USD 110 In-stock
Estimated Time of Arrival: December 31
200 mg USD 190 In-stock
Estimated Time of Arrival: December 31
500 mg USD 340 In-stock
Estimated Time of Arrival: December 31
1 g   Get quote  
5 g   Get quote  

* Please select Quantity before adding items.

Customer Review

Other Forms of Piribedil:

  • Biological Activity

  • Technical Information

  • Purity & Documentation

  • References

Description

Piribedil is a dopamine D2 receptor (D2R) agonist which also displays antagonist property at 1A-adrenoceptor (1A-AR).

IC50 & Target

D2R, hα1A-AR[1]

Clinical Trial
Solvent & Solubility
In Vitro: 

DMSO : 33.33 mg/mL (111.72 mM; Need ultrasonic)

Preparing
Stock Solutions
Concentration Solvent Mass 1 mg 5 mg 10 mg
1 mM 3.3519 mL 16.7594 mL 33.5188 mL
5 mM 0.6704 mL 3.3519 mL 6.7038 mL
10 mM 0.3352 mL 1.6759 mL 3.3519 mL
*Please refer to the solubility information to select the appropriate solvent.
In Vivo:
  • 1.

    Add each solvent one by one:  10% DMSO    90% corn oil

    Solubility: ≥ 2.5 mg/mL (8.38 mM); Clear solution

  • 2.

    Add each solvent one by one:  10% DMSO    40% PEG300    5% Tween-80    45% saline

    Solubility: ≥ 2.5 mg/mL (8.38 mM); Clear solution

  • 3.

    Add each solvent one by one:  10% DMSO    90% (20% SBE-β-CD in saline)

    Solubility: ≥ 2.5 mg/mL (8.38 mM); Clear solution

References
Molecular Weight

298.34

Formula

C₁₆H₁₈N₄O₂

CAS No.

3605-01-4

SMILES

C1(N2CCN(CC3=CC=C(OCO4)C4=C3)CC2)=NC=CC=N1

Storage
Powder -20°C 3 years
  4°C 2 years
In solvent -80°C 6 months
  -20°C 1 month
Shipping

Room temperature in continental US; may vary elsewhere

  • Molarity Calculator

  • Dilution Calculator

The molarity calculator equation

Mass (g) = Concentration (mol/L) × Volume (L) × Molecular Weight (g/mol)

Mass   Concentration   Volume   Molecular Weight *
= × ×

The dilution calculator equation

Concentration (start) × Volume (start) = Concentration (final) × Volume (final)

This equation is commonly abbreviated as: C1V1 = C2V2

Concentration (start) × Volume (start) = Concentration (final) × Volume (final)
× = ×
C1   V1   C2   V2

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Product Name:
Piribedil
Cat. No.:
HY-12707
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Piribedil

Cat. No.: HY-12707