LPAR5 Modulator
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LPAR5 Modulator (1)
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N-PTyrosine PA ammonium
0 ImagesCat. No.: HY-W040176CAS No.: 799268-45-4Synonyms: N-Palmitoyl-tyrosine phosphoric acid ammoniumN-PTyrosine PA (N-Palmitoyl-tyrosine phosphoric acid) ammonium is a lysophosphatidic acid (LPA) receptor modulator, which exhibits weak inhibitory activity against LPA1 and partial agonist properties towards LPA5. N-PTyrosine PA ammonium inhibits the activation of LPA receptors and downstream responses by competing with agonists for binding sites. N-PTyrosine PA ammonium can induce morphological changes and aggregation, and also inhibit LPA-induced morphological changes through receptor desensitization caused by pre-incubation. N-PTyrosine PA ammonium can be used in the research of related diseases such as atherosclerosis and acute ischemic syndromes (e.g., unstable angina, myocardial infarction, stroke).
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August 31
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August 31
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