Amylin agonist 1
Amylin agonist 1 is an agonist of amylin receptor 3 (AMY3R), with an EC50 of 6.17 nM for stimulating cellular cAMP production. Amylin agonist 1 is also an agonist of calcitonin receptor (CTR), with an EC50 of 8.58 nM. Amylin agonist 1 can be used for the research of type 2 diabetes and obesity.
For research use only. We do not sell to patients.
- Formula: C33H37ClN8O4
- Molecular Weight:645.15
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Storage:
Please store the product under the recommended conditions in the Certificate of Analysis.
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Biological Activity
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Chemical Information
- Purity & Documentation
- References
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Help & FAQs
Biological Activity
Amylin agonist 1 (Example 239a) potently activates the amylin 3 receptor, with a relative EC50 of 6.17 nM and an Emax of 105%[1].
Amylin agonist 1 potently activates the calcitonin receptor, with a relative EC50 of 8.58 nM and an Emax of 96%[1].
MedChemExpress (MCE) has not independently confirmed the accuracy of these methods. They are for reference only.
Chemical Information
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Molecular Weight 645.15
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Formula C33H37ClN8O4
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SMILES
CC(CC1=C(C(C2=CC=C3C(OCC(N3CC4=NC=C(C=N4)Cl)=O)=C2)=C5C=NN(C5=N1)C6CCN(CC6C)C7COC7)C(N)=O)C
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Shipping
Room temperature in continental US; may vary elsewhere.
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Storage
Please store the product under the recommended conditions in the Certificate of Analysis.
Purity & Documentation
References
Calculators
Concentration (start) × Volume (start) = Concentration (final) × Volume (final)
Amylin agonist 1 Related Classifications
HY-179728 Related Classifications
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