TD-6301
TD-6301 is a bladder-selective M2/4 muscarinic receptor antagonist. TD-6301 binds to and blocks M2/4 muscarinic receptors with high selectivity, especially human M2 receptors with strong affinity (Ki = 0.36 nM). TD-6301 inhibits volume-induced bladder contractions (ID50 = 0.075 mg/kg). TD-6301 can be used in the research of overactive bladder.
Nur für Forschungszwecke. Wir verkaufen nicht an Patienten.
- CAS. Nr.: 690999-15-6
- Formel: C40H57N5O2
- Molecular Weight:639.91
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Speicherung:
Please store the product under the recommended conditions in the Certificate of Analysis.
Biologische Aktivität
Ki: 0.36 nM (human M2 muscarinic receptor)
Chemical Information
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CAS. Nr. 690999-15-6
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Molecular Weight 639.91
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Formel C40H57N5O2
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SMILES
NC(C(C1=CC=CC=C1)(C2=CC=CC=C2)[C@H]3CN(CC3)CCCCCCCN(C4CCN(CC4)CC5=CN=CC=C5OC)C(C)C)=O
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Versand
Room temperature in continental US; may vary elsewhere.
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Speicherung
Please store the product under the recommended conditions in the Certificate of Analysis.
Reinheit & Dokumentation
Verweise
Calculators
Konzentration (Stammlösung) × Volumen (Stammlösung) = Konzentration (Ziellösung) × Volumen (Ziellösung)