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Cat. No.: HY-172095

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BRD4 Inhibitor-39

BRD4 Inhibitor-39 (compound 12m) is an orally available BRD4 inhibitor with an IC₅₀ value of 0.02 μM. BRD4 Inhibitor-39 induces apoptosis. BRD4 Inhibitor-39 has anti-tumor activity.

For research use only. We do not sell to patients.

CAS No.: 3069926-33-3
Formula: C₂₄H₁₉BrFN₉
Molecular Weight:532.37

Storage:

Please store the product under the recommended conditions in the Certificate of Analysis.

Data Sheet (270 KB)

BRD4 Inhibitor-39 Chemical Structure

CAS No.: 3069926-33-3

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Use of MCE Products

Strong Fluorescence Signal / Multi-Disciplinary Applications / High Fluorescence Specificity

Biological Activity

Description

BRD4 Inhibitor-39 (compound 12m) is an orally available BRD4 inhibitor with an IC₅₀ value of 0.02 μM. BRD4 Inhibitor-39 induces apoptosis. BRD4 Inhibitor-39 has anti-tumor activity^[1].

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Chemical Information

CAS No. 3069926-33-3
Molecular Weight 532.37
Formula C₂₄H₁₉BrFN₉
SMILES

FC1=CC(Br)=C(C=C1)NC2=C(N=C3N2C=C(N=C3)C4=CN(N=C4)C)C(C=C5)=CN6C5=NN=C6CC
Shipping

Room temperature in continental US; may vary elsewhere.
Storage

Please store the product under the recommended conditions in the Certificate of Analysis.

Purity & Documentation

Select Batch:

Purity: 99.98%

Assay: 99.98%

ee.: 99.98%

Data Sheet (270 KB)
COA (2659 KB)
Elemental Analysis Report (2659 KB)
HNMR (2659 KB)
CNMR (2659 KB)
RP-HPLC (2659 KB)
NP-HPLC (2659 KB)
MS (2659 KB)
LCMS (2659 KB)
IR (2659 KB)
GC (2659 KB)
OR (2659 KB)
SDS-PAGE (2659 KB)
SEC-HPLC (2659 KB)
Other Report (2659 KB)
Handling Instructions (2659 KB)

References

[1]. Liu JY, et al. Design, synthesis, and antitumor evaluation of triazolopyridine derivatives as novel inhibitors for BRD4. Eur J Med Chem. 2025 Jan 13;285:117272. [Content Brief]

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Help & FAQs

How should lyophilized recombinant proteins be reconstituted and stored?

1. Before opening the cap, centrifuge the vial at 13000 rpm for 20-30 seconds. This step will ensure that any lyophilized powder that may have adhered to the cap or walls is collected at the bottom of the vial, minimizing the risk of product loss.

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Chemical Information
Purity & Documentation
References

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BRD4 Inhibitor-39

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