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Cat. No.: HY-153660S

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Bivamelagon-d₈

Name: Bivamelagon-d8
Brand: MedChemExpress
SKU: HY-153660S
Availability: PreOrder

(Synonyms: MC-4R Agonist 2-d₈)

Bivamelagon-d₈ (MC-4R Agonist 2-d₈) is the deuterium labeled Bivamelagon (HY-153660). Bivamelagon (MC-4R Agonist 2) is an orally active MC4R agonist with EC₅₀ values of 0.562 nM (Luci assay) and 36.5 nM (cAMP assay), and a K_i of 65 nM. Bivamelagon can be used for the research of diseases such as obesity and diabetes.

Nos produits utilisent uniquement pour la recherche. Nous ne vendons pas aux patients.

Formule: C₃₅H₄₅D₈ClN₄O₄
Masse moléculaire:637.32

Stockage:

Please store the product under the recommended conditions in the Certificate of Analysis.

Bivamelagon-d₈ Chemical Structure

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Activité biologique
- Description
- In Vitro
- Application
Chemical Information
Pureté et documentation
Calculators
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Bioz

Activité biologique

Description

Voir tous les produits spécifiques à Isoform Melanocortin Receptor :

In Vitro

Stable heavy isotopes of hydrogen, carbon, and other elements have been incorporated into drug molecules, largely as tracers for quantitation during the drug development process. Deuteration has gained attention because of its potential to affect the pharmacokinetic and metabolic profiles of drugs.

MedChemExpress (MCE) has not independently confirmed the accuracy of these methods. They are for reference only.

Application

1. This compound can be used as a tracer
2. This compound can be used as an internal standard for quantitative analysis by NMR, GC-MS, or LC-MS.

Chemical Information

Unlabeled CAS 2641595-54-0
Masse moléculaire 637.32
Formule C₃₅H₄₅D₈ClN₄O₄
SMILES

O=C([C@H]1[C@H](C2=CC=C(C=C2)Cl)CN(C1)C(C)(C)C)N3[C@@H](C[C@@H](C3)N([C@@H]4CC[C@@H](CC4)C)C(C(C)C)=O)C(N5C([2H])([2H])C([2H])([2H])OC([2H])([2H])C5([2H])[2H])=O
Synonyms

MC-4R Agonist 2-d₈
Livraison

Room temperature in continental US; may vary elsewhere.
Stockage

Please store the product under the recommended conditions in the Certificate of Analysis.