LM-030
LM-030 (BPR277), cyclic depsipeptide, is a potent kallikrein-related peptidase 7 (KLK7) and human neutrophil elastase inhibitor with IC50 values of 1 and 10 nM. LM-030 can be used for the study of Netherton syndrome.
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- CAS No.: 1122484-55-2
- Formule: C46H72N8O12
- Masse moléculaire:929.11
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Stockage:
Please store the product under the recommended conditions in the Certificate of Analysis.
Activité biologique
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KLK7 1 nM (IC50) |
| NCT Number | Sponsor | Condition | Start Date |
Phase
|
|---|---|---|---|---|
| NCT01329991 | Plexxikon| | 2011-05 | PHASE1 |
Chemical Information
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CAS No. 1122484-55-2
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Masse moléculaire 929.11
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Formule C46H72N8O12
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Synonyms
BPR277
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Sequence
Gln-lactone[Thr-Leu-{Oaa}-Tyr-Ile]
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Sequence Shortening
Q-lactone[TL-{Oaa}-YI]
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Livraison
Room temperature in continental US; may vary elsewhere.
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Stockage
Please store the product under the recommended conditions in the Certificate of Analysis.
Pureté et documentation
Références
Calculators
Concentration (start) × Volume (start) = Concentration (final) × Volume (final)