SSTR4 agonist 5
SSTR4 agonist 5 (Compound 5) is the orally active agonist for somatostatin receptor 4 (SSTR4) with an EC50 of 0.228 nM. SSTR4 agonist 5 exhibits good stability in human/rat liver microsomes. SSTR4 agonist 5 inhibits mechanical hyperalgesia in rat models.
Nos produits utilisent uniquement pour la recherche. Nous ne vendons pas aux patients.
- CAS No.: 2761347-44-6
- Formule: C20H26N4O
- Masse moléculaire:338.45
-
Stockage:
Please store the product under the recommended conditions in the Certificate of Analysis.
Activité biologique
Description
IC50 & Target
|
SSTR4 0.228 nM (IC50) |
Chemical Information
-
CAS No. 2761347-44-6
-
Masse moléculaire 338.45
-
Formule C20H26N4O
-
SMILES
O=C(C1C2CNCC12C)NC(C)(C)C3=NC4=C5C(CCC4)=CC=CN35
-
Livraison
Room temperature in continental US; may vary elsewhere.
-
Stockage
Please store the product under the recommended conditions in the Certificate of Analysis.
Pureté et documentation
Références
Calculators
Concentration (start) × Volume (start) = Concentration (final) × Volume (final)