102704-40-5
102704-40-5
Chemical Structure
GAT211
- CAS No.: 102704-40-5
- Formula:C22H18N2O2
- Molecular Weight:342.39
IUPAC Name: 3-(2-nitro-1-phenylethyl)-2-phenyl-1H-indole
InChIKey: OHZDCJJHWPHZJD-UHFFFAOYSA-N
SMILES: O=[N+]([O-])CC(C1=CC=CC=C1)C2=C(NC3=C2C=CC=C3)C4=CC=CC=C4
Biological Activity: GAT211 is a cannabinoid 1 receptor (CB1R) positive allosteric modulator (PAM). GAT211 activates cAMP and β-arrestin2 with EC50 values of 260 nM and 650 nM, respectively. GAT211 inhibits GAT211 can be used for neuropathic and/or inflammatory pain research[1].
| Cat. No. | Product Name | Purity | Description | Pricing | |||||||||||||||||||
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GAT211 | 99.96% | GAT211 is a cannabinoid 1 receptor (CB1R) positive allosteric modulator (PAM). GAT211 activates cAMP and β-arrestin2 with EC50 values of 260 nM and 650 nM, respectively. GAT211 inhibits GAT211 can be used for neuropathic and/or inflammatory pain research. | ||||||||||||||||||||
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Structural Analogs
-
Similarity Score 1.00
HY-120953GAT228 -
Similarity Score 1.00
HY-121600GAT229 -
Similarity Score 0.83
HY-150056CB1R Allosteric modulator 3 -
Similarity Score 0.81
HY-144705GAT564 -
Similarity Score 0.68
HY-118140ZCZ011 -
Similarity Score 0.64
HY-150057CB1R Allosteric modulator 4 -
Similarity Score 0.56
HY-15722SB-222200 -
Similarity Score 0.55
HY-150407TSPO ligand-1 -
Similarity Score 0.54
HY-143250Tubulin inhibitor 12 -
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