108437-87-2
![[D-Phe12]-Bombesin Chemical Structure](http://file.medchemexpress.cn/product_pic/hy-103282.gif "[D-Phe12]-Bombesin Chemical Structure")
Chemical Structure
[D-Phe12]-Bombesin
- CAS No.: 108437-87-2
- Formula:C74H112N22O18S
- Molecular Weight:1629.88
IUPAC Name: (S)-N1-((5S,8S,11R,17S,20S,23S,26S,29S,35S,38S)-23-((1H-indol-3-yl)methyl)-43-amino-29-(2-amino-2-oxoethyl)-26-(3-amino-3-oxopropyl)-11-benzyl-5-carbamoyl-43-imino-8,35-diisobutyl-17-isopropyl-20-methyl-7,10,13,16,19,22,25,28,31,34,37-undecaoxo-2-thia-6,9
InChIKey: NXZVGUQLNAVPLJ-VKXSZNMLSA-N
SMILES: O=C([C@@H](N1)CCC1=O)N[C@@H](CCC(N)=O)C(N[C@@H](CCCNC(N)=N)C(N[C@@H](CC(C)C)C(NCC(N[C@@H](CC(N)=O)C(N[C@@H](CCC(N)=O)C(N[C@H](C(N[C@@H](C)C(N[C@@H](C(C)C)C(NCC(N[C@@H](C(N[C@@H](CC(C)C)C(N[C@H](C(N)=O)CCSC)=O)=O)CC2=CC=CC=C2)=O)=O)=O)=O)CC3=CNC4=C3C=CC=C4)=O)=O)=O)=O)=O)=O
Biological Activity: [D-Phe12]-Bombesin is a derivative of Bombesin (HY-P0195) and an antagonist for bombesin receptor with Ki of 4.7 μM. [D-Phe12]-Bombesin inhibits the Bombesin (HY-P0195)-induced amylase release, with IC50 of 4 μM[1].
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[D-Phe12]-Bombesin | [D-Phe12]-Bombesin is a derivative of Bombesin (HY-P0195) and an antagonist for bombesin receptor with Ki of 4.7 μM. [D-Phe12]-Bombesin inhibits the Bombesin (HY-P0195)-induced amylase release, with IC50 of 4 μM. | |||||||||||||||||||||
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Keywords
