1176326-76-3
1176326-76-3
Chemical Structure
DSP-1053
- CAS No.: 1176326-76-3
- Formula:C26H32BrNO4
- Molecular Weight:502.44
IUPAC Name: 6-(2-(4-(4-bromo-3-(2-methoxyethoxy)benzyl)piperidin-1-yl)ethyl)chroman-4-one
InChIKey: ZSVLGHSNQJYODD-UHFFFAOYSA-N
SMILES: BrC1=CC=C(CC2CCN(CCC3=CC(C(CCO4)=O)=C4C=C3)CC2)C=C1OCCOC
Biological Activity: DSP-1053, a benzylpiperidine derivative, is a potent Serotonin Transporter (SERT) inhibitor with a Ki of 1.02 nM. DSP-1053 shows partial 5-HT1A receptor agonistic activity with a Ki of 5.05 nM. DSP-1053 has antidepressant activity[1].
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DSP-1053 | 99.75% | DSP-1053, a benzylpiperidine derivative, is a potent Serotonin Transporter (SERT) inhibitor with a Ki of 1.02 nM. DSP-1053 shows partial 5-HT1A receptor agonistic activity with a Ki of 5.05 nM. DSP-1053 has antidepressant activity. | ||||||||||||||||||||
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DSP-1053 (Standard) | ≥98% | DSP-1053 (Standard) is the analytical standard of DSP-1053 (HY-111419). This product is intended for research and analytical applications. DSP-1053, a benzylpiperidine derivative, is a potent Serotonin Transporter (SERT) inhibitor with a Ki of 1.02 nM. DSP-1053 shows partial 5-HT1A receptor agonistic activity with a Ki of 5.05 nM. DSP-1053 has antidepressant activity. | ||||||||||||||||||||
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Structural Analogs
-
Similarity Score 0.82
HY-111419ADSP-1053 benzenesulfonate -
Similarity Score 0.51
HY-151562AChE/BuChE/MAO-B-IN-1 -
Similarity Score 0.51
HY-101815Lidanserin -
Similarity Score 0.49
HY-117774AHR-2244 hydrochloride -
Similarity Score 0.49
HY-W747696Donepezil impurity 11 hydrochloride -
Similarity Score 0.49
HY-B0034RDonepezil Hydrochloride (Standard) -
Similarity Score 0.49
HY-13510Cutamesine dihydrochloride -
Similarity Score 0.49
HY-W747696ADonepezil impurity 11 -
Similarity Score 0.49
HY-14940Volinanserin -
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