AChE/BuChE/MAO-B-IN-1
AChE/BuChE/MAO-B-IN-1 (compound 19) is an inhibitor of human acetyl- (hAChE), butyrylcholinesterase (hBuChE) and monoamine oxidase-B (hMAO-B) with IC50s of 4.8 μM, 13.7 μM, and 1.11 μM, respectively. AChE/BuChE/MAO-B-IN-1 also exhibits high affinity to both the σ1 and σ2 receptors with Ki values of 42.8 nM (human σ1 receptor) and 191 nM (rat σ2 receptor), respectively. AChE/BuChE/MAO-B-IN-1 can be used for Alzheimer’s disease research.
For research use only. We do not sell to patients.
- CAS No.: 2834758-29-9
- Formula: C17H23NO3
- Molecular Weight:289.37
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Storage:
Please store the product under the recommended conditions in the Certificate of Analysis.
To place orders, for customer services and technical support, please contact: MedChemExpress USA
Tel: 609-228-6898 E-mail: [email protected] [email protected]
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Biological Activity
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Chemical Information
- Purity & Documentation
- References
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Help & FAQs
Biological Activity
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hAChE 4.8 μM (IC50) |
hBCHE 13.7 μM (IC50) |
hMAO-B 1.11 μM (IC50) |
Chemical Information
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CAS No. 2834758-29-9
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Molecular Weight 289.37
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Formula C17H23NO3
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SMILES
O=C1CCOC2=C1C=C(OCCN3CCCCCC3)C=C2
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Shipping
Room temperature in continental US; may vary elsewhere.
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Storage
Please store the product under the recommended conditions in the Certificate of Analysis.
Purity & Documentation
References
Calculators
Concentration (start) × Volume (start) = Concentration (final) × Volume (final)
AChE/BuChE/MAO-B-IN-1 Related Classifications
HY-151562 Related Classifications
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