1228182-44-2
1228182-44-2
Chemical Structure
Cimaterol-d7
Synonym(s): CL 263780-d7
- CAS No.: 1228182-44-2
- Formula:C12H10D7N3O
- Molecular Weight:226.33
IUPAC Name: 2-amino-5-(1-hydroxy-2-((propan-2-yl-d7)amino)ethyl)benzonitrile
InChIKey: BUXRLJCGHZZYNE-UNAVHCQLSA-N
SMILES: N#CC1=CC(C(O)CNC(C([2H])([2H])[2H])([2H])C([2H])([2H])[2H])=CC=C1N
Biological Activity: Cimaterol-d7 is the deuterium labeled Cimaterol. Cimaterol is a potent agonist of β-adrenergic receptors (pEC50s=8.13, 8.78, and 6.62 for human β1, β2, and β3, respectively). Cimaterol has been used in farmed animals to increase carcass mass and to alter muscle and fat deposition.
| Cat. No. | Product Name | Purity | Description | Pricing | |||||||||||||||||||
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
|
|
Cimaterol-d7 | Cimaterol-d7 is the deuterium labeled Cimaterol. Cimaterol is a potent agonist of β-adrenergic receptors (pEC50s=8.13, 8.78, and 6.62 for human β1, β2, and β3, respectively). Cimaterol has been used in farmed animals to increase carcass mass and to alter muscle and fat deposition. | |||||||||||||||||||||
|
loading...
/
|
|||||||||||||||||||||||
|
|
Cimaterol (Standard) | ≥98% | Cimaterol (Standard) is the analytical standard of Cimaterol. This product is intended for research and analytical applications. Cimaterol (CL 263780) is a β-adrenergic agonist on energy metabolism in ob/ob mice. The Kd for Cimaterol binding to the L6 β-receptor is 26 nM which is compatible with its EC50 for the stimulation of protein synthesis (approx 5 nM). | ||||||||||||||||||||
|
loading...
/
|
|||||||||||||||||||||||
|
|
Cimaterol | 99.13% | Cimaterol (CL 263780) is a β-adrenergic agonist on energy metabolism in ob/ob mice. The Kd for Cimaterol binding to the L6 β-receptor is 26 nM which is compatible with its EC50 for the stimulation of protein synthesis (approx 5 nM). | ||||||||||||||||||||
|
loading...
/
|
|||||||||||||||||||||||
