1334107-58-2
1334107-58-2
Chemical Structure
Akt1&PKA-IN-1
- CAS No.: 1334107-58-2
- Formula:C20H17Cl2N3O
- Molecular Weight:386.27
IUPAC Name: (S)-N-(azetidin-3-yl(3,4-dichlorophenyl)methyl)isoquinoline-6-carboxamide
InChIKey: TWAIYMKBHKNSRO-LJQANCHMSA-N
SMILES: O=C(C1=CC2=C(C=NC=C2)C=C1)N[C@@H](C3CNC3)C4=CC(Cl)=C(C=C4)Cl
Biological Activity: Akt1&PKA-IN-1 is a potent dual Akt/PKA inhibitor with IC50 values of 0.03 , 0.11 μM, and 9.8 μM for PKAa, Akt, and CDK2, respectively. Akt1&PKA-IN-1 is selective for cyclin-dependent kinase 2 (CDK2)[1].
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Akt1&PKA-IN-1 | Akt1&PKA-IN-1 is a potent dual Akt/PKA inhibitor with IC50 values of 0.03 , 0.11 μM, and 9.8 μM for PKAa, Akt, and CDK2, respectively. Akt1&PKA-IN-1 is selective for cyclin-dependent kinase 2 (CDK2). | |||||||||||||||||||||
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References
Keywords
