Akt1&PKA-IN-1
Akt1&PKA-IN-1 is a potent dual Akt/PKA inhibitor with IC50 values of 0.03 , 0.11 μM, and 9.8 μM for PKAa, Akt, and CDK2, respectively. Akt1&PKA-IN-1 is selective for cyclin-dependent kinase 2 (CDK2).
For research use only. We do not sell to patients.
- CAS No.: 1334107-58-2
- Formula: C20H17Cl2N3O
- Molecular Weight:386.27
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Storage:
Please store the product under the recommended conditions in the Certificate of Analysis.
Biological Activity
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PKAa 0.03 μM (IC50) |
Akt 0.11 μM (IC50) |
CDK2 9.8 μM (IC50) |
Chemical Information
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CAS No. 1334107-58-2
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Molecular Weight 386.27
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Formula C20H17Cl2N3O
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SMILES
O=C(C1=CC2=C(C=NC=C2)C=C1)N[C@@H](C3CNC3)C4=CC(Cl)=C(C=C4)Cl
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Shipping
Room temperature in continental US; may vary elsewhere.
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Storage
Please store the product under the recommended conditions in the Certificate of Analysis.
Purity & Documentation
References
Calculators
Concentration (start) × Volume (start) = Concentration (final) × Volume (final)