1346572-63-1
Chemical Structure
GSK503
- CAS No.: 1346572-63-1
- Formula:C31H38N6O2
- Molecular Weight:526.67
IUPAC Name: N-((4,6-dimethyl-2-oxo-1,2-dihydropyridin-3-yl)methyl)-1-isopropyl-3-methyl-6-(6-(4-methylpiperazin-1-yl)pyridin-3-yl)-1H-indole-4-carboxamide
InChIKey: HRDQQHUKUIKFHT-UHFFFAOYSA-N
SMILES: O=C(C1=CC(C2=CC=C(N3CCN(C)CC3)N=C2)=CC4=C1C(C)=CN4C(C)C)NCC5=C(C)C=C(C)NC5=O
Biological Activity: GSK503 is a potent and specific inhibitor of EZH2 methyltransferase with Kiapp values of 3 to 27 nM.
| Cat. No. | 상품명 | Purity | 제품 설명 | Pricing | |||||||||||||||||||
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
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GSK503 | 99.52% | GSK503 is a potent and specific inhibitor of EZH2 methyltransferase with Kiapp values of 3 to 27 nM. | ||||||||||||||||||||
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-
Similarity Score 0.85
HY-13470GSK126 -
Similarity Score 0.79
HY-116605GSK926 -
Similarity Score 0.75
HY-148458EZH2-IN-14 -
Similarity Score 0.73
HY-W1063360EZH2 ligand-5 -
Similarity Score 0.69
HY-15646UNC1999 -
Similarity Score 0.66
HY-13500GSK343 -
Similarity Score 0.65
HY-181393EZH2 ligand-3 -
Similarity Score 0.64
HY-100846RJQEZ5 (Standard) -
Similarity Score 0.61
HY-133129MS1943 -
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