1346574-57-9
1346574-57-9
Chemical Structure
GSK126
Synonym(s): GSK2816126A
- CAS No.: 1346574-57-9
- Formula:C31H38N6O2
- Molecular Weight:526.67
IUPAC Name: (S)-1-(sec-butyl)-N-((4,6-dimethyl-2-oxo-1,2-dihydropyridin-3-yl)methyl)-3-methyl-6-(6-(piperazin-1-yl)pyridin-3-yl)-1H-indole-4-carboxamide
InChIKey: FKSFKBQGSFSOSM-QFIPXVFZSA-N
SMILES: O=C(C1=CC(C2=CC=C(N3CCNCC3)N=C2)=CC4=C1C(C)=CN4[C@@H](C)CC)NCC5=C(C)C=C(C)NC5=O
Biological Activity: GSK126 (GSK2816126A) is a potent, highly selective inhibitor of EZH2 methyltransferase with an IC50 of 9.9 nM[1].
| Cat. No. | Product Name | Purity | Description | Pricing | |||||||||||||||||||
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GSK126 | 99.75% | GSK126 (GSK2816126A) is a potent, highly selective inhibitor of EZH2 methyltransferase with an IC50 of 9.9 nM. | ||||||||||||||||||||
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References
Keywords
