1620107-33-6
1620107-33-6
Chemical Structure
LU-005i
- CAS No.: 1620107-33-6
- Formula:C31H46N4O7
- Molecular Weight:586.72
IUPAC Name: (S)-N-((S)-3-cyclohexyl-1-((R)-2-methyloxiran-2-yl)-1-oxopropan-2-yl)-3-(4-methoxyphenyl)-2-((S)-2-(2-morpholinoacetamido)propanamido)propanamide
InChIKey: UHNYITHLNFUAIN-VTNASVEKSA-N
SMILES: COC(C=C1)=CC=C1C[C@H](NC([C@H](C)NC(CN2CCOCC2)=O)=O)C(N[C@@H](CC3CCCCC3)C([C@]4(CO4)C)=O)=O
Biological Activity: LU-005i is a potent inhibitor of β5i subunit of immunoproteasomes (IC50 = 6.6 nM), selective over β5c subunit (IC50 = 287 nM)[1].
| Cat. No. | Product Name | Purity | Description | Pricing | |||||||||||||||||||
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
|
|
LU-005i | 98.24% | LU-005i is a potent inhibitor of β5i subunit of immunoproteasomes (IC50 = 6.6 nM), selective over β5c subunit (IC50 = 287 nM). | ||||||||||||||||||||
|
loading...
/
|
|||||||||||||||||||||||
References
Keywords
