168079-32-1
168079-32-1
Chemical Structure
Lixivaptan
Synonym(s): VPA-985; WAY-VPA 985
- CAS No.: 168079-32-1
- Formula:C27H21ClFN3O2
- Molecular Weight:473.93
IUPAC Name: N-(3-chloro-4-(10,11-dihydro-5H-benzo[e]pyrrolo[1,2-a][1,4]diazepine-10-carbonyl)phenyl)-5-fluoro-2-methylbenzamide
InChIKey: PPHTXRNHTVLQED-UHFFFAOYSA-N
SMILES: O=C(C1=C(Cl)C=C(NC(C2=CC(F)=CC=C2C)=O)C=C1)N(C3)C4=CC=CC=C4CN5C3=CC=C5
Biological Activity: Lixivaptan (VPA-985, WAY-VPA 985) is an orally active and selective vasopressin receptor V2 antagonist, with IC50 values of 1.2 and 2.3 nM for human and rat V2, respectively.
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Lixivaptan | 99.67% | Lixivaptan (VPA-985, WAY-VPA 985) is an orally active and selective vasopressin receptor V2 antagonist, with IC50 values of 1.2 and 2.3 nM for human and rat V2, respectively. | ||||||||||||||||||||
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Lixivaptan (Standard) | ≥98% | Lixivaptan (Standard) is the analytical standard of Lixivaptan. This product is intended for research and analytical applications. Lixivaptan (VPA-985, WAY-VPA 985) is an orally active and selective vasopressin receptor V2 antagonist, with IC50 values of 1.2 and 2.3 nM for human and rat V2, respectively. | ||||||||||||||||||||
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Keywords
