2020052-55-3

CDK12-IN-E9 Chemical Structure
2020052-55-3

Chemical Structure

CDK12-IN-E9

  • CAS No.: 2020052-55-3
  • Formula:C24H30N6O2
  • Molecular Weight:434.53

IUPAC Name: (S)-N-(3-((3-ethyl-5-(2-(2-hydroxyethyl)piperidin-1-yl)pyrazolo[1,5-a]pyrimidin-7-yl)amino)phenyl)acrylamide

InChIKey: CDCHESFKYUNJPV-FQEVSTJZSA-N

SMILES: C=CC(NC1=CC=CC(NC2=CC(N3[C@H](CCO)CCCC3)=NC4=C(CC)C=NN24)=C1)=O

Biological Activity: CDK12-IN-E9 is a potent and selective covalent CDK12 inhibitor and a non-covalent CDK9 inhibitor, while avoiding ABC transporter-mediated efflux. CDK12-IN-E9 has weak binding ability to CDK7/CyclinH complex with an IC50> 1 μM[1].

Cat. No. Product Name Purity Description Pricing
HY-117203A 		CDK12-IN-E9 99.71% CDK12-IN-E9 is a potent and selective covalent CDK12 inhibitor and a non-covalent CDK9 inhibitor, while avoiding ABC transporter-mediated efflux. CDK12-IN-E9 has weak binding ability to CDK7/CyclinH complex with an IC50> 1 μM.
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