217438-17-0
Chemical Structure
SB 268262
- CAS No.: 217438-17-0
- Formula:C18H15N3O4S2
- Molecular Weight:401.46
IUPAC Name: N-methyl-3-nitro-4-(thiazol-2-ylsulfinyl)-N-(o-tolyl)benzamide
InChIKey: YXHLPJQQPOMPGE-UHFFFAOYSA-N
SMILES: O=C(N(C)C1=CC=CC=C1C)C2=CC=C(S(C3=NC=CS3)=O)C([N+]([O-])=O)=C2
Biological Activity: CGRP antagonist 4 is an antagonist of calcitonin gene-related peptide (CGRP) receptor. CGRP antagonist 4 shows the highest affinity for CGRP receptors in the human brain. CGRP antagonist 4 can be used to study the binding properties of non-peptide calcitonin gene-related peptide (CGRP) receptor antagonist (gepants) in rat, pig and human menes [1].
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SB 268262 | 99.9% | CGRP antagonist 4 is an antagonist of calcitonin gene-related peptide (CGRP) receptor. CGRP antagonist 4 shows the highest affinity for CGRP receptors in the human brain. CGRP antagonist 4 can be used to study the binding properties of non-peptide calcitonin gene-related peptide (CGRP) receptor antagonist (gepants) in rat, pig and human menes . | ||||||||||||||||||||
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Keywords