2245255-65-4
2245255-65-4
Chemical Structure
GSK2807
- CAS No.: 2245255-65-4
- Formula:C19H32N8O5
- Molecular Weight:452.51
IUPAC Name: (S)-2-amino-4-((((2R,3S,4R,5R)-5-(6-amino-9H-purin-9-yl)-3,4-dihydroxytetrahydrofuran-2-yl)methyl)(3-(dimethylamino)propyl)amino)butanoic acid
InChIKey: FYXRZDCUJHGULY-URQYDQELSA-N
SMILES: NC1=C(N=CN2[C@@H]3O[C@H](CN(CC[C@H](N)C(O)=O)CCCN(C)C)[C@@H](O)[C@H]3O)C2=NC=N1
Biological Activity: GSK2807 is a potent and selective SAM-competitive inhibitor of SMYD3, exhibiting a Ki value of 14 nM, and it may be useful for cancer treatment by preventing the methylation of MEKK2.
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GSK2807 | GSK2807 is a potent and selective SAM-competitive inhibitor of SMYD3, exhibiting a Ki value of 14 nM, and it may be useful for cancer treatment by preventing the methylation of MEKK2. | |||||||||||||||||||||
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Keywords
