2259641-24-0
2259641-24-0
Chemical Structure
Ep300/CREBBP-IN-8
- CAS No.: 2259641-24-0
- Formula:C25H27F2N5O3
- Molecular Weight:483.51
IUPAC Name: (2R,4R)-4-fluoro-1-(1-(3-fluoro-4-methoxyphenyl)cyclohexane-1-carbonyl)-N-(1H-pyrazolo[4,3-b]pyridin-5-yl)pyrrolidine-2-carboxamide
InChIKey: IQSXIRMYLOUTLS-OXQOHEQNSA-N
SMILES: O=C([C@@H]1N(C(C2(C3=CC=C(OC)C(F)=C3)CCCCC2)=O)C[C@H](F)C1)NC4=CC=C(NN=C5)C5=N4
Biological Activity: Ep300/CREBBP-IN-8 (Example 37) is a potent and orally active Ep300 and CREBBP inhibitor with IC50s of 0.014 and 0.018 μM, respectively. Ep300/CREBBP-IN-8 can be used for the research of cancer[1].
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Ep300/CREBBP-IN-8 | Ep300/CREBBP-IN-8 (Example 37) is a potent and orally active Ep300 and CREBBP inhibitor with IC50s of 0.014 and 0.018 μM, respectively. Ep300/CREBBP-IN-8 can be used for the research of cancer. | |||||||||||||||||||||
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References
Keywords
