2408841-19-8
2408841-19-8
Chemical Structure
PKM2-IN-3
- CAS No.: 2408841-19-8
- Formula:C21H22O4
- Molecular Weight:338.40
IUPAC Name: (E)-4-(4-ethylbenzylidene)-6,8-dimethoxy-3,4-dihydrobenzo[b]oxepin-5(2H)-one
InChIKey: BQNYBXFXLMWECE-LFIBNONCSA-N
SMILES: COC1=C2C(OCC/C(C2=O)=C\C3=CC=C(C=C3)CC)=CC(OC)=C1
Biological Activity: PKM2-IN-3 is an inhibitor of PKM2 kinase with an IC50 value of 4.1 μM. PKM2-IN-3 exhibits an anti-neuroinflammatory effect by inhibiting PKM2-mediated glycolysis and NLRP3 activation[1].
| Cat. No. | Product Name | Purity | Description | Pricing | |||||||||||||||||||
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
|
|
PKM2-IN-3 | 99.44% | PKM2-IN-3 is an inhibitor of PKM2 kinase with an IC50 value of 4.1 μM. PKM2-IN-3 exhibits an anti-neuroinflammatory effect by inhibiting PKM2-mediated glycolysis and NLRP3 activation. | ||||||||||||||||||||
|
loading...
/
|
|||||||||||||||||||||||
References
Keywords
