2535970-65-9
Chemical Structure
EST73502 monohydrochloride
- CAS No.: 2535970-65-9
- Formula:C19H27ClF2N2O2
- Molecular Weight:388.88
IUPAC Name: (R)-9-(2,5-difluorophenethyl)-4-ethyl-2-methyl-1-oxa-4,9-diazaspiro[5.5]undecan-3-one hydrochloride
InChIKey: WZJJIHSIBMZUIN-PFEQFJNWSA-N
SMILES: FC1=CC=C(F)C=C1CCN(CC2)CCC2(O[C@@H]3C)CN(CC)C3=O.[H]Cl
Biological Activity: EST73502 monohydrochloride is a selective, orally active and blood-brain barrier (BBB) penetrant dual μ-opioid receptor (MOR) agonist and σ1 receptor (σ1R) antagonist, with Kis of 64 nM and 118 nM for MOR and σ1R, respectively. EST73502 monohydrochloride has antinociceptive activity[1].
| Cat. No. | Product Name | Purity | Description | Pricing | |||||||||||||||||||
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EST73502 monohydrochloride | 99.58% | EST73502 monohydrochloride is a selective, orally active and blood-brain barrier (BBB) penetrant dual μ-opioid receptor (MOR) agonist and σ1 receptor (σ1R) antagonist, with Kis of 64 nM and 118 nM for MOR and σ1R, respectively. EST73502 monohydrochloride has antinociceptive activity. | ||||||||||||||||||||
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Keywords
