2755890-53-8
Chemical Structure
PF-07258669
- CAS No.: 2755890-53-8
- Formula:C25H27FN6O2
- Molecular Weight:462.52
IUPAC Name: (R)-2-(5-fluoro-2-methoxypyridin-4-yl)-1-((S)-7'-methyl-6'-(pyrimidin-2-yl)-3',4'-dihydro-1'H-spiro[pyrrolidine-3,2'-[1,8]naphthyridin]-1-yl)propan-1-one
InChIKey: PARGFYLSRQUWHR-BZQUYTCOSA-N
SMILES: CC(N=C(N1)C(CC[C@]21CCN(C([C@H](C)C3=C(C=NC(OC)=C3)F)=O)C2)=C4)=C4C5=NC=CC=N5
Biological Activity: PF-07258669 is an orally active melanocortin-4 receptor (MC4R) antagonist that antagonizes MC4R with an IC50 of 13 nM (Ki=0.46 nM). PF-07258669 can be used for the research of cachexia, anorexia, or anorexia nervosa[1].
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PF-07258669 | 98.46% | PF-07258669 is an orally active melanocortin-4 receptor (MC4R) antagonist that antagonizes MC4R with an IC50 of 13 nM (Ki=0.46 nM). PF-07258669 can be used for the research of cachexia, anorexia, or anorexia nervosa. | ||||||||||||||||||||
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Keywords
