2828567-39-9
2828567-39-9
Chemical Structure
Rentosertib
Synonym(s): INS018_055; TNIK&MAP4K4-IN-2
- CAS No.: 2828567-39-9
- Formula:C27H30FN7O
- Molecular Weight:487.57
InChIKey: ZVDNXHUSIKGTSF-UHFFFAOYSA-N
SMILES: O=C(C1=CN=C(C2=C(C3=CC=C(C=C3)F)N=CN2C(C)C)N1)NC4=CC=C(N5CCN(CC5)C)C=C4
Biological Activity: Rentosertib (INS018 055) (compound 112) is the orally active TNIK and MAP4K4 inhibitor with IC50 values of 12-120, 12-120 nM, respectively[1].
| Cat. No. | Product Name | Purity | Description | Pricing | |||||||||||||||||||
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Rentosertib | 99.96% | Rentosertib (INS018 055) (compound 112) is the orally active TNIK and MAP4K4 inhibitor with IC50 values of 12-120, 12-120 nM, respectively. | ||||||||||||||||||||
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Structural Analogs
-
Similarity Score 0.53
HY-151292Antitumor agent-74 -
Similarity Score 0.53
HY-151295Antitumor agent-75 -
Similarity Score 0.53
HY-149262CLK1-IN-3 -
Similarity Score 0.53
HY-145044HPK1-IN-17 -
Similarity Score 0.52
HY-146262LDC0496 -
Similarity Score 0.52
HY-184315LDC8201 -
Similarity Score 0.51
HY-156523TNIK&MAP4K4-IN-1 -
Similarity Score 0.51
HY-100794GR127935 hydrochloride -
Similarity Score 0.51
HY-123869GR127935 -
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