2847829-86-9

PROTAC ER Degrader-16 Chemical Structure
2847829-86-9

Chemical Structure

PROTAC ER Degrader-16

  • CAS No.: 2847829-86-9
  • Formula:C47H54BN5O6
  • Molecular Weight:795.77

InChIKey: KNJAMZGBBBEBDI-INXUWUOZSA-N

SMILES: CC/C(C1=CC=CC=C1)=C(C2=CC=C(C=C2)B(O)O)/C3=CC=C(C=C3)OCCN4CCN(CC4)CC5CCN(CC5)C6=CC7=C(C(N(C7)C8CCC(NC8=O)=O)=O)C=C6

Biological Activity: PROTAC ER Degrader-16 is an orally active ERα PROTAC degrader with a DC50 of 1.4 nM and an IC50 of 1.9 nM. PROTAC ER Degrader-16 inhibits ER-dependent breast cancer cell proliferation and exerts anti-tumor effects in mouse models. PROTAC ER Degrader-16 can be used for breast cancer research[1].

Cat. No. Product Name Purity Description Pricing
HY-183804 		PROTAC ER Degrader-16 PROTAC ER Degrader-16 is an orally active ERα PROTAC degrader with a DC50 of 1.4 nM and an IC50 of 1.9 nM. PROTAC ER Degrader-16 inhibits ER-dependent breast cancer cell proliferation and exerts anti-tumor effects in mouse models. PROTAC ER Degrader-16 can be used for breast cancer research.
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