287206-61-5
Chemical Structure
MA-2029
- CAS No.: 287206-61-5
- Formula:C31H45FN4O4
- Molecular Weight:556.71
IUPAC Name: (S)-N-((S)-3-(3-(tert-butyl)-4-hydroxyphenyl)-1-(ethylamino)-1-oxopropan-2-yl)-2-((S)-3-(4-fluorophenyl)-N-methyl-2-(methylamino)propanamido)-3-methylbutanamide
InChIKey: KSDWAJPUTRBIRR-KLJDGLGGSA-N
SMILES: FC(C=C1)=CC=C1C[C@H](NC)C(N(C)[C@@H](C(C)C)C(N[C@H](C(NCC)=O)CC2=CC(C(C)(C)C)=C(O)C=C2)=O)=O
Biological Activity: MA-2029 is a selective, orally active, and competitive motilin receptor antagonist (IC50=4.9 nM). MA-2029 is selective for the motilin receptor over various other receptors and ion channels. MA-2029 may be useful for gastrointestinal disorders associated with disturbed gastrointestinal motility[1].
| Cat. No. | Product Name | Purity | Description | Pricing | |||||||||||||||||||
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MA-2029 | 98.94% | MA-2029 is a selective, orally active, and competitive motilin receptor antagonist (IC50=4.9 nM). MA-2029 is selective for the motilin receptor over various other receptors and ion channels. MA-2029 may be useful for gastrointestinal disorders associated with disturbed gastrointestinal motility. | ||||||||||||||||||||
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Keywords
