2910938-59-7
Chemical Structure
CK156
- CAS No.: 2910938-59-7
- Formula:C21H25N5O3
- Molecular Weight:395.45
IUPAC Name: (13Z,14E)-N-(tert-butyl)-3,6-dioxa-9-aza-1(3,5)-pyrazolo[1,5-a]pyrimidina-2(1,3)-benzenacyclononaphane-24-carboxamide
InChIKey: YCFFONJEHNSECY-UHFFFAOYSA-N
SMILES: O=C(C1=CC=C2C=C1OCCOCCNC3=NC4=C2C=NN4C=C3)NC(C)(C)C
Biological Activity: CK156, a chemical probe, is a highly selective death-associated protein kinase (DAPK) inhibitor with IC50s of 182 nM,34 μM, and 39 μM in the DRAK1 NanoBRET assay for DRAK1, CK2a1, and CK2a2, respectively. CK156 can be used for the research of autoimmune and inflammatory diseases[1].
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CK156 | 99.60% | CK156, a chemical probe, is a highly selective death-associated protein kinase (DAPK) inhibitor with IC50s of 182 nM,34 μM, and 39 μM in the DRAK1 NanoBRET assay for DRAK1, CK2a1, and CK2a2, respectively. CK156 can be used for the research of autoimmune and inflammatory diseases. | ||||||||||||||||||||
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Keywords
