4929-23-1
4929-23-1
Chemical Structure
BI-0115
- CAS No.: 4929-23-1
- Formula:C15H14ClN3O
- Molecular Weight:287.74
IUPAC Name: 9-chloro-5-propyl-5,11-dihydro-6H-benzo[e]pyrido[3,2-b][1,4]diazepin-6-one
InChIKey: QTCZUCSALXBZQR-UHFFFAOYSA-N
SMILES: O=C1N(CCC)C2=CC=CN=C2NC3=CC(Cl)=CC=C13
Biological Activity: BI-0115 is a selective inhibitor of LOX-1 (IC50=5.4 μM) that blocks cellular uptake of oxLDL. BI-0115 binding triggers receptor inhibition by formation of dimers of the homodimeric ligand binding domain[1].
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BI-0115 | 99.72% | BI-0115 is a selective inhibitor of LOX-1 (IC50=5.4 μM) that blocks cellular uptake of oxLDL. BI-0115 binding triggers receptor inhibition by formation of dimers of the homodimeric ligand binding domain. | ||||||||||||||||||||
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References
Keywords
