515141-51-2
515141-51-2
Chemical Structure
GW-803430
Synonym(s): GW-3430
- CAS No.: 515141-51-2
- Formula:C25H24ClN3O3S
- Molecular Weight:481.99
IUPAC Name: 6-(4-chlorophenyl)-3-(3-methoxy-4-(2-(pyrrolidin-1-yl)ethoxy)phenyl)thieno[3,2-d]pyrimidin-4(3H)-one
InChIKey: MWULMTACIBZPGN-UHFFFAOYSA-N
SMILES: O=C1C2=C(C=C(C3=CC=C(Cl)C=C3)S2)N=CN1C4=CC=C(OCCN5CCCC5)C(OC)=C4
Biological Activity: GW-803430 (GW-3430) is a potent and selective melanin-concentrating hormone receptor 1 (MCH R1) antagonist with a pIC50 of 9.3. GW-803430 is orally active in an animal model of obesity[1].
| Cat. No. | Product Name | Purity | Description | Pricing | |||||||||||||||||||
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GW-803430 | 98.53% | GW-803430 (GW-3430) is a potent and selective melanin-concentrating hormone receptor 1 (MCH R1) antagonist with a pIC50 of 9.3. GW-803430 is orally active in an animal model of obesity. | ||||||||||||||||||||
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GW-803430 (Standard) | ≥98% | GW-803430 (Standard) is the analytical standard of GW-803430 (HY-11083). This product is intended for research and analytical applications. GW-803430 (GW-3430) is a potent and selective melanin-concentrating hormone receptor 1 (MCH R1) antagonist with a pIC50 of 9.3. GW-803430 is orally active in an animal model of obesity. | ||||||||||||||||||||
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Structural Analogs
-
Similarity Score 0.80
HY-12433BMS-819881 -
Similarity Score 0.77
HY-120608BMS-814580 -
Similarity Score 0.74
HY-12433ABMS-830216 -
Similarity Score 0.72
HY-108049GW856464 -
Similarity Score 0.51
HY-Z8379Raloxifene impurity 4 -
Similarity Score 0.51
HY-135590Raloxifene 4-Monomethyl Ether -
Similarity Score 0.51
HY-135584Raloxifene 6-Monomethyl Ether -
Similarity Score 0.50
HY-116896RLY117018 (Standard) -
Similarity Score 0.50
HY-135580ARaloxifene Bismethyl Ether hydrochloride -
Explore the MedChemAI to find more analogs
