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  3. Raloxifene 6-Monomethyl Ether

Raloxifene 6-Monomethyl Ether 

Cat. No.: HY-135584
Handling Instructions

Raloxifene 6-Monomethyl Ether (Compound 7) is a Raloxifene derivative that inhibits estrogen receptor α. Raloxifene 4-Monomethyl Ether inhibits MCF-7 cells with an IC50 of 250 nM and a pIC50 of 6.6.

For research use only. We do not sell to patients.

Raloxifene 6-Monomethyl Ether Chemical Structure

Raloxifene 6-Monomethyl Ether Chemical Structure

CAS No. : 178451-13-3

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Description

Raloxifene 6-Monomethyl Ether (Compound 7) is a Raloxifene derivative that inhibits estrogen receptor α. Raloxifene 4-Monomethyl Ether inhibits MCF-7 cells with an IC50 of 250 nM and a pIC50 of 6.6[1].

In Vitro

Raloxifene 6-Monomethyl Ether (Compound 7) is a Raloxifene derivative with a methoxy group on C6. Raloxifene 6-Monomethyl Ether holds poor ICsub>50 value because of disruption to the hydrogen bond network and steric disfavor[1].

Molecular Weight

487.61

Formula

C₂₉H₂₉NO₄S

CAS No.

178451-13-3

SMILES

O=C(C1=C(C2=CC=C(O)C=C2)SC3=CC(OC)=CC=C31)C4=CC=C(OCCN5CCCCC5)C=C4

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Room temperature in continental US; may vary elsewhere.

Storage

Please store the product under the recommended conditions in the Certificate of Analysis.

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Keywords:

Raloxifene 6-Monomethyl EtherEstrogen Receptor/ERRERαRaloxifenederivativemethoxyInhibitorinhibitorinhibit

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Raloxifene 6-Monomethyl Ether
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HY-135584
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