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Cat. No.: HY-12433A

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BMS-830216

BMS-830216 is an antagonist of MCHR-1. BMS-830216 is a phosphate ester prodrug. BMS-830216 can be studied in obesity-related research.

For research use only. We do not sell to patients.

CAS No.: 1197420-06-6
Formula: C₂₄H₂₂ClN₂O₇PS
Molecular Weight:548.93

Storage:

Please store the product under the recommended conditions in the Certificate of Analysis.

Data Sheet (265 KB)

BMS-830216 Chemical Structure

CAS No.: 1197420-06-6

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Use of MCE Products

Fluorescent Dye

Strong Fluorescence Signal / Multi-Disciplinary Applications / High Fluorescence Specificity

Biological Activity
- Description
- Clinical Trial
Chemical Information
Purity & Documentation
References
Calculators
Help & FAQs
Classifications
Bioz

Biological Activity

Description

BMS-830216 is an antagonist of MCHR-1. BMS-830216 is a phosphate ester prodrug. BMS-830216 can be studied in obesity-related research^[1].

Clinical Trial

NCT Number	Sponsor	Condition	Start Date	Phase A549
NCT01329991	Plexxikon\|		2011-05	PHASE1

Chemical Information

CAS No. 1197420-06-6
Molecular Weight 548.93
Formula C₂₄H₂₂ClN₂O₇PS
SMILES

ClC1=CC=C(C2=CC(N=CN(C3=CC(OC)=C(OC[C@H](OP(O)(O)=O)C4CC4)C=C3)C5=O)=C5S2)C=C1
Shipping

Room temperature in continental US; may vary elsewhere.
Storage

Please store the product under the recommended conditions in the Certificate of Analysis.

Purity & Documentation

Select Batch:

Purity: 99.98%

Assay: 99.98%

ee.: 99.98%

Data Sheet (265 KB)
COA (2659 KB)
Elemental Analysis Report (2659 KB)
HNMR (2659 KB)
CNMR (2659 KB)
RP-HPLC (2659 KB)
NP-HPLC (2659 KB)
MS (2659 KB)
LCMS (2659 KB)
IR (2659 KB)
GC (2659 KB)
OR (2659 KB)
SDS-PAGE (2659 KB)
SEC-HPLC (2659 KB)
Other Report (2659 KB)
Handling Instructions (2659 KB)

References

[1]. Washburn, W. N., et al., (2014). Identification of a nonbasic melanin hormone receptor 1 antagonist as an antiobesity clinical candidate. Journal of medicinal chemistry, 57(18), 7509-7522. [Content Brief]

Calculators

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Help & FAQs

How should lyophilized recombinant proteins be reconstituted and stored?

1. Before opening the cap, centrifuge the vial at 13000 rpm for 20-30 seconds. This step will ensure that any lyophilized powder that may have adhered to the cap or walls is collected at the bottom of the vial, minimizing the risk of product loss.

Keywords

100 mg

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