54765-26-3
54765-26-3
Chemical Structure
Lerimazoline
- CAS No.: 54765-26-3
- Formula:C13H18N2
- Molecular Weight:202.30
IUPAC Name: 2-(2,4,6-trimethylbenzyl)-4,5-dihydro-1H-imidazole
InChIKey: DUHARNKZLBMPBS-UHFFFAOYSA-N
SMILES: CC1=C(CC2=NCCN2)C(C)=CC(C)=C1
Biological Activity: Lerimazoline is a selective 5-HT1D receptor agonist with Ki values of 72 and 3480 nM for h5-HT1D and h5-HT1B. Lerimazoline inhibits Forskolin (HY-15371)-stimulated cAMP production and induces contractions in rabbit saphenous vein preparations. Lerimazoline can be used for the research of migraine[1].
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Lerimazoline | Lerimazoline is a selective 5-HT1D receptor agonist with Ki values of 72 and 3480 nM for h5-HT1D and h5-HT1B. Lerimazoline inhibits Forskolin (HY-15371)-stimulated cAMP production and induces contractions in rabbit saphenous vein preparations. Lerimazoline can be used for the research of migraine. | |||||||||||||||||||||
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References
Keywords
