82857-38-3
Chemical Structure
Bopindolol malonate
Synonym(s): (±)-Bopindolol malonate
- CAS No.: 82857-38-3
- Formula:C26H32N2O7
- Molecular Weight:484.54
IUPAC Name: 1-(tert-butylamino)-3-((2-methyl-1H-indol-4-yl)oxy)propan-2-yl benzoate malonate
InChIKey: LDOONRJGLKHGJI-UHFFFAOYSA-N
SMILES: CC(N1)=CC2=C1C=CC=C2OCC(OC(C3=CC=CC=C3)=O)CNC(C)(C)C.O=C(O)CC(O)=O
Biological Activity: Bopindolol ((±)-Bopindolol) malonate is an orally active antagonist of β-adrenoceptors (ARs) with partial agonist activity. Bopindolol malonate is non-selective for β1- and β2-ARs and has low affinity for β3-AR subtype. Bopindolol malonate has intrinsic sympathomimetic as well as membrane stabilizing actions, inhibits renin secretion, and interacts with 5-HT receptors. Bopindolol malonate is a proagent of Pindolol (HY-B0982). Bopindolol malonate can be used for essential and renovascular hypertension research.
| Cat. No. | Product Name | Purity | Description | Pricing | |||||||||||||||||||
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Bopindolol malonate | 98.3% | Bopindolol ((±)-Bopindolol) malonate is an orally active antagonist of β-adrenoceptors (ARs) with partial agonist activity. Bopindolol malonate is non-selective for β1- and β2-ARs and has low affinity for β3-AR subtype. Bopindolol malonate has intrinsic sympathomimetic as well as membrane stabilizing actions, inhibits renin secretion, and interacts with 5-HT receptors. Bopindolol malonate is a proagent of Pindolol (HY-B0982). Bopindolol malonate can be used for essential and renovascular hypertension research. | ||||||||||||||||||||
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Keywords
