CGP 54626 hydrochloride

Art. -Nr.: HY-101378 Reinheit: 99.76%: Data Sheet
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Handling Instructions
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CGP 54626 (hydrochloride) is a selective antagonist of GABA_B receptor with an IC₅₀ value of 4 nM. CGP 54626 (hydrochloride) can be used to investigate the role of GABA_B receptors in neurological signaling.

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CGP 54626 hydrochloride Chemische Struktur

CAS. Nr. : 149184-21-4

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1 mg	Auf Lager	Estimated Time of Arrival: December 31
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10 mg	Angebot einholen

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This product is a controlled substance and not for sale in your territory.

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Based on 2 publication(s) in Google Scholar

Other Forms of CGP 54626 hydrochloride:

CGP 54626 Angebot einholen

2 Publications Citing Use of MCE CGP 54626 hydrochloride

Spezialitätsempfehlungen

•Related Screening Libraries:

•Related Small Molecules:

•Related Proteins:

Biologische Aktivität
Reinheit & Dokumentation
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Beschreibung

Cellular Effect

Cell Line	Type	Value	Description	References
CHO	IC₅₀	6.4 nM Compound: CGP-54626	Displacement of [3H]CGP54626 from human recombinant GABAB1A receptor expressed in CHO cells after 3 hrs Displacement of [3H]CGP54626 from human recombinant GABAB1A receptor expressed in CHO cells after 3 hrs	[PMID: 23403082]

Molekulargewicht

444.76

Formel

C₁₈H₂₉Cl₃NO₃P

CAS. Nr.

149184-21-4

Appearance

Solid

Color

White to off-white

SMILES

O=P(C[C@@H](O)CN[C@H](C1=CC=C(Cl)C(Cl)=C1)C)(CC2CCCCC2)O.Cl

Versand

Room temperature in continental US; may vary elsewhere.

Speicherung

-20°C, protect from light, stored under nitrogen

*In solvent : -80°C, 6 months; -20°C, 1 month (protect from light, stored under nitrogen)

Reinheit & Dokumentation

Purity: 99.76%

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Data Sheet (266 KB) SDS (252 KB)

COA (246 KB) LCMS (88 KB)

Handling Instructions (2659 KB)

Verweise

[1]. Kaupmann K, et al. GABA(B)-receptor subtypes assemble into functional heteromeric complexes. Nature. 1998 Dec 17;396(6712):683-7. [Content Brief]