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Art. -Nr.: HY-147343

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P300-IN-2

P300-IN-2 is a p300 inhibitor (IC₅₀=3.6 μM) that inhibits histone acetyltransferase p300 activity. P300-IN-2 shows weak inhibitory activity against CWR22RV1 cell proliferation. P300-IN-2 can be used for research on p300-mediated diseases, such as cancer.

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CAS. Nr.: 2488867-43-0
Formel: C₂₆H₂₇FN₄O₅
Molecular Weight:494.52

Speicherung:

Please store the product under the recommended conditions in the Certificate of Analysis.

P300-IN-2 Chemical Structure

CAS. Nr.: 2488867-43-0

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Use of MCE Products

Strong Fluorescence Signal / Multi-Disciplinary Applications / High Fluorescence Specificity

Biologische Aktivität
- Beschreibung
- IC₅₀ & Target
- In Vitro
Chemical Information
Reinheit & Dokumentation
Verweise
Calculators
Help & FAQs
Classifications
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Biologische Aktivität

Beschreibung

IC₅₀ & Target

^[1]

p300

3.6 μM (IC₅₀)

Alle Histone Acetyltransferase Isoform-spezifische Produkte anzeigen :

In Vitro

P300-IN-2 (compound 17) shows weak inhibitory activity against CWR22RV1 cell proliferation, with an IC₅₀ > 2000 nM^[1].

P300-IN-2 inhibits the histone acetyltransferase p300 with an IC₅₀ of 3.6 μM^[1].

MedChemExpress (MCE) has not independently confirmed the accuracy of these methods. They are for reference only.

Related Protocols :

Chemical Information

CAS. Nr. 2488867-43-0
Molecular Weight 494.52
Formel C₂₆H₂₇FN₄O₅
SMILES

O=C1[C@@]2(C=3C(CC2)=CC(NC(NC)=O)=CC3)OC(=O)N1CC(=O)N4[C@H](CC[C@H]4C)C5=CC=C(F)C=C5
Versand

Room temperature in continental US; may vary elsewhere.
Speicherung

Please store the product under the recommended conditions in the Certificate of Analysis.

Reinheit & Dokumentation

Handling Instructions (2659 KB)

Verweise

[1]. Fan L, et al. Histone acetylase p300 inhibitor and application thereof. CN111217802A, 2020.

Calculators

Molaritätsrechner

Mass (g) = Concentration (mol/L) × Volume (L) × Molecular Weight (g/mol)

Mass Mass

Konzentration Konzentration

Volumen Volumen

Molecular Weight Molecular Weight

Verdünnungsrechner

Konzentration _{(Stammlösung)} × Volumen _{(Stammlösung)} = Konzentration _{(Ziellösung)} × Volumen _{(Ziellösung)}

Konzentration _{(Stammlösung)} Konzentration _{(Stammlösung)}

Volumen _{(Stammlösung)} Volumen _{(Stammlösung)}

Konzentration _{(Ziellösung)} Konzentration _{(Ziellösung)}

Volumen _{(Ziellösung)} Volumen _{(Ziellösung)}

Help & FAQs

How should lyophilized recombinant proteins be reconstituted and stored?

1. Before opening the cap, centrifuge the vial at 13000 rpm for 20-30 seconds. This step will ensure that any lyophilized powder that may have adhered to the cap or walls is collected at the bottom of the vial, minimizing the risk of product loss.

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100 mg

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Biologische Aktivität
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- In Vitro
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P300-IN-2

Alle Histone Acetyltransferase Isoform-spezifische Produkte anzeigen

Biologische Aktivität

Beschreibung

IC50 & Target

In Vitro

Chemical Information

Reinheit & Dokumentation

Verweise

Calculators

Help & FAQs

P300-IN-2 Related Classifications

HY-147343 Related Classifications

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