LPE-1
LPE-1 is a lysine-specific demethylase 1 (LSD1) inhibitor with an IC50 of 0.65 μM. LPE-1 inhibits the proliferation of gastric cancer, liver cancer and prostate cancer cells, and shows no activity against a subset of gastric cancer cells. LPE-1 is applicable for the research of gastric cancer, liver cancer and prostate cancer.
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- CAS No.: 1637373-70-6
- Formule: C13H10N6S3
- Masse moléculaire:346.45
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Stockage:
Please store the product under the recommended conditions in the Certificate of Analysis.
To place orders, for customer services and technical support, please contact: MedChemExpress USA
Tel: 609-228-6898 E-mail: [email protected] [email protected]
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Activité biologique
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Chemical Information
- Pureté et documentation
- Références
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Help & FAQs
Activité biologique
LPE-1 (Compound Ⅰ-12) (72 h) inhibits the proliferation of MGC-803 (IC50 = 7.85 μM), HGC-27 (IC50 = 5.16 μM), HepG2 (IC50 = 5.71 μM) and PC-3 (IC50 = 7.21 μM) cells, but shows no detectable activity against SGC-7901 cells (IC50 >128 μM)[1].
MedChemExpress (MCE) has not independently confirmed the accuracy of these methods. They are for reference only.
Chemical Information
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CAS No. 1637373-70-6
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Masse moléculaire 346.45
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Formule C13H10N6S3
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SMILES
N#CC=1C(=NC(=NC1C=2SC=CC2)SCC#C)NNC(=S)N
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Livraison
Room temperature in continental US; may vary elsewhere.
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Stockage
Please store the product under the recommended conditions in the Certificate of Analysis.
Pureté et documentation
Références
Calculators
Concentration (start) × Volume (start) = Concentration (final) × Volume (final)
LPE-1 Related Classifications
HY-155825 Related Classifications
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