1. GPCR/G Protein
    Neuronal Signaling
  2. 5-HT Receptor
  3. Cisapride monohydrate

Cisapride monohydrate (Synonyms: R 51619 monohydrate; (±)-Cisaprid monohydrate)

Cat. No.: HY-14149A
Handling Instructions

Cisapride monohydrate is an orally and potent 5-HT4 receptor agonist and hERG inhibitor. Cisapride monohydrate is an prokinetic agent which facilitates or restores motility throughout the length of the gastrointestinal tract. Cisapride monohydrate stimulates gastrointestinal motor activity through an indirect mechanism involving the release of acetylcholine mediated by postganglionic nerve endings in the myenteric plexus of the gut.

For research use only. We do not sell to patients.

Cisapride monohydrate Chemical Structure

Cisapride monohydrate Chemical Structure

CAS No. : 260779-88-2

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Description

Cisapride monohydrate is an orally and potent 5-HT4 receptor agonist and hERG inhibitor. Cisapride monohydrate is an prokinetic agent which facilitates or restores motility throughout the length of the gastrointestinal tract. Cisapride monohydrate stimulates gastrointestinal motor activity through an indirect mechanism involving the release of acetylcholine mediated by postganglionic nerve endings in the myenteric plexus of the gut[1][2].

IC50 & Target

5-HT4 Receptor

0.14 μM (EC50)

Molecular Weight

483.96

Formula

C23H31ClFN3O5

CAS No.
SMILES

ClC1=C(N)C=C(OC)C(C(N[[email protected]]2[[email protected]@H](OC)CN(CCCOC3=CC=C(F)C=C3)CC2)=O)=C1.O

Shipping

Room temperature in continental US; may vary elsewhere.

Storage

Please store the product under the recommended conditions in the Certificate of Analysis.

Purity & Documentation
References
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Product Name:
Cisapride monohydrate
Cat. No.:
HY-14149A
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