Dopamine D3 receptor ligand-5
Dopamine D3 receptor ligand-5 (13a), a Cariprazine (HY-14763) analogue, is a dopamine D3 receptor ligand, with Ki values of 2.85 nM and 0.14 nM for D2R and D3R, respectively.
For research use only. We do not sell to patients.
- CAS No.: 2899250-94-1
- Formula: C22H33Cl2N3O2
- Molecular Weight:442.42
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Storage:
Please store the product under the recommended conditions in the Certificate of Analysis.
Biological Activity
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D3 Receptor 0.14 nM (Ki) |
5-HT2B Receptor 1.47 nM (Ki) |
D2 Receptor 2.85 nM (Ki) |
5-HT1A Receptor 6 nM (Ki) |
5-HT2A Receptor 54 nM (Ki) |
5-HT2C Receptor 252 nM (Ki) |
D4 Receptor 756 nM (Ki) |
D1 Receptor 4600 nM (Ki) |
MedChemExpress (MCE) has not independently confirmed the accuracy of these methods. They are for reference only.
Chemical Information
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CAS No. 2899250-94-1
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Molecular Weight 442.42
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Formula C22H33Cl2N3O2
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SMILES
ClC1=C(C=CC=C1Cl)N2CCN(CC2)CC[C@@H]3CC[C@H](CC3)NC(CCOC)=O
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Shipping
Room temperature in continental US; may vary elsewhere.
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Storage
Please store the product under the recommended conditions in the Certificate of Analysis.
Purity & Documentation
References
Calculators
Concentration (start) × Volume (start) = Concentration (final) × Volume (final)