SSTR4 agonist 5
SSTR4 agonist 5 (Compound 5) is the orally active agonist for somatostatin receptor 4 (SSTR4) with an EC50 of 0.228 nM. SSTR4 agonist 5 exhibits good stability in human/rat liver microsomes. SSTR4 agonist 5 inhibits mechanical hyperalgesia in rat models.
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- No. CAS: 2761347-44-6
- Fòrmula: C20H26N4O
- Peso molecular:338.45
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Almacenamiento:
Please store the product under the recommended conditions in the Certificate of Analysis.
Actividad biológica
Descripciòn
IC50 & Target
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SSTR4 0.228 nM (IC50) |
Chemical Information
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No. CAS 2761347-44-6
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Peso molecular 338.45
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Fòrmula C20H26N4O
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SMILES
O=C(C1C2CNCC12C)NC(C)(C)C3=NC4=C5C(CCC4)=CC=CN35
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Envío
Room temperature in continental US; may vary elsewhere.
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Almacenamiento
Please store the product under the recommended conditions in the Certificate of Analysis.
Pureza y Documentación
Referencias
Calculators
Concentration (start) × Volume (start) = Concentration (final) × Volume (final)