LPE-1
LPE-1 is a lysine-specific demethylase 1 (LSD1) inhibitor with an IC50 of 0.65 μM. LPE-1 inhibits the proliferation of gastric cancer, liver cancer and prostate cancer cells, and shows no activity against a subset of gastric cancer cells. LPE-1 is applicable for the research of gastric cancer, liver cancer and prostate cancer.
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- No. CAS: 1637373-70-6
- Fòrmula: C13H10N6S3
- Peso molecular:346.45
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Almacenamiento:
Please store the product under the recommended conditions in the Certificate of Analysis.
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Actividad biológica
Descripciòn
In Vitro
LPE-1 (Compound Ⅰ-12) (72 h) inhibits the proliferation of MGC-803 (IC50 = 7.85 μM), HGC-27 (IC50 = 5.16 μM), HepG2 (IC50 = 5.71 μM) and PC-3 (IC50 = 7.21 μM) cells, but shows no detectable activity against SGC-7901 cells (IC50 >128 μM)[1].
MedChemExpress (MCE) has not independently confirmed the accuracy of these methods. They are for reference only.
Chemical Information
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No. CAS 1637373-70-6
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Peso molecular 346.45
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Fòrmula C13H10N6S3
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SMILES
N#CC=1C(=NC(=NC1C=2SC=CC2)SCC#C)NNC(=S)N
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Envío
Room temperature in continental US; may vary elsewhere.
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Almacenamiento
Please store the product under the recommended conditions in the Certificate of Analysis.
Pureza y Documentación
Referencias
Calculators
Concentration (start) × Volume (start) = Concentration (final) × Volume (final)
LPE-1 Related Classifications
HY-155825 Related Classifications
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