1. GPCR/G Protein
  2. GnRH Receptor
  3. GnRH antagonist 2

GnRH antagonist 2 (formula I) is a GnRH receptor antagonist that can be used for endometriosis research.

For research use only. We do not sell to patients.

GnRH antagonist 2 Chemical Structure

GnRH antagonist 2 Chemical Structure

CAS No. : 1709823-61-9

Size Price Stock Quantity
Solid + Solvent
10 mM * 1 mL in DMSO
ready for reconstitution
USD 668 In-stock
Solution
10 mM * 1 mL in DMSO USD 668 In-stock
Solid
5 mg USD 500 In-stock
10 mg USD 850 In-stock
25 mg USD 1800 In-stock
50 mg USD 3000 In-stock
100 mg   Get quote  
200 mg   Get quote  

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Based on 1 publication(s) in Google Scholar

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Description

GnRH antagonist 2 (formula I) is a GnRH receptor antagonist that can be used for endometriosis research[1].

Molecular Weight

607.57

Formula

C28H27F2N9O5

CAS No.
Appearance

Solid

Color

White to yellow

SMILES

O=C(NOC)NC1=CC=C(N2N=C(C(C(N3C4=NN=C(OC)C=C4)=O)=C2CN(C)C)N(CC5=C(F)C=CC=C5F)C3=O)C=C1

Shipping

Room temperature in continental US; may vary elsewhere.

Storage
Powder -20°C 3 years
4°C 2 years
In solvent -80°C 6 months
-20°C 1 month
Solvent & Solubility
In Vitro: 

DMSO : 150 mg/mL (246.89 mM; ultrasonic and warming and heat to 60°C; Hygroscopic DMSO has a significant impact on the solubility of product, please use newly opened DMSO)

Preparing
Stock Solutions
Concentration Solvent Mass 1 mg 5 mg 10 mg
1 mM 1.6459 mL 8.2295 mL 16.4590 mL
5 mM 0.3292 mL 1.6459 mL 3.2918 mL
View the Complete Stock Solution Preparation Table

* Please refer to the solubility information to select the appropriate solvent. Once prepared, please aliquot and store the solution to prevent product inactivation from repeated freeze-thaw cycles.
Storage method and period of stock solution: -80°C, 6 months; -20°C, 1 month. When stored at -80°C, please use it within 6 months. When stored at -20°C, please use it within 1 month.

  • Molarity Calculator

  • Dilution Calculator

Mass (g) = Concentration (mol/L) × Volume (L) × Molecular Weight (g/mol)

Mass
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Concentration
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Volume
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Molecular Weight *

Concentration (start) × Volume (start) = Concentration (final) × Volume (final)

This equation is commonly abbreviated as: C1V1 = C2V2

Concentration (start)

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Volume (start)

V1

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Concentration (final)

C2

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Volume (final)

V2

In Vivo Dissolution Calculator
Please enter the basic information of animal experiments:

Dosage

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g

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(per animal)

μL

Number of animals

Recommended: Prepare an additional quantity of animals to account for potential losses during experiments.
Calculation results:
Working solution concentration: mg/mL
Purity & Documentation

Purity: 98.16%

References

Complete Stock Solution Preparation Table

* Please refer to the solubility information to select the appropriate solvent. Once prepared, please aliquot and store the solution to prevent product inactivation from repeated freeze-thaw cycles.
Storage method and period of stock solution: -80°C, 6 months; -20°C, 1 month. When stored at -80°C, please use it within 6 months. When stored at -20°C, please use it within 1 month.

Optional Solvent Concentration Solvent Mass 1 mg 5 mg 10 mg 25 mg
DMSO 1 mM 1.6459 mL 8.2295 mL 16.4590 mL 41.1475 mL
5 mM 0.3292 mL 1.6459 mL 3.2918 mL 8.2295 mL
10 mM 0.1646 mL 0.8230 mL 1.6459 mL 4.1148 mL
15 mM 0.1097 mL 0.5486 mL 1.0973 mL 2.7432 mL
20 mM 0.0823 mL 0.4115 mL 0.8230 mL 2.0574 mL
25 mM 0.0658 mL 0.3292 mL 0.6584 mL 1.6459 mL
30 mM 0.0549 mL 0.2743 mL 0.5486 mL 1.3716 mL
40 mM 0.0411 mL 0.2057 mL 0.4115 mL 1.0287 mL
50 mM 0.0329 mL 0.1646 mL 0.3292 mL 0.8230 mL
60 mM 0.0274 mL 0.1372 mL 0.2743 mL 0.6858 mL
80 mM 0.0206 mL 0.1029 mL 0.2057 mL 0.5143 mL
100 mM 0.0165 mL 0.0823 mL 0.1646 mL 0.4115 mL
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GnRH antagonist 2 Related Classifications

Help & FAQs
  • Do most proteins show cross-species activity?

    Species cross-reactivity must be investigated individually for each product. Many human cytokines will produce a nice response in mouse cell lines, and many mouse proteins will show activity on human cells. Other proteins may have a lower specific activity when used in the opposite species.

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Product Name:
GnRH antagonist 2
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HY-134864
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