2. GPCR/G Protein Neuronal Signaling
  3. Cannabinoid Receptor
  4. GP1a

GP1a is a potent agonist of cannabinoid receptor 2 (CB2). Gp1a is beneficial to skin wound healing. GP1a inhibits inflammation and fibrogenesis while promoting re-epithelialization.

For research use only. We do not sell to patients.

GP1a Chemical Structure

GP1a Chemical Structure

CAS No. : 511532-96-0

Size Price Stock Quantity
1 mg USD 65 In-stock
5 mg USD 140 In-stock
10 mg USD 220 In-stock
25 mg USD 435 In-stock
50 mg   Get quote  
100 mg   Get quote  

* Please select Quantity before adding items.

This product is a controlled substance and not for sale in your territory.

Customer Review

Based on 1 publication(s) in Google Scholar

GP1a Related Antibodies

Top Publications Citing Use of Products

View All Cannabinoid Receptor Isoform Specific Products:

View All Isoforms

  • Biological Activity

  • Purity & Documentation

  • References

  • Customer Review

Description

GP1a is a potent agonist of cannabinoid receptor 2 (CB2). Gp1a is beneficial to skin wound healing. GP1a inhibits inflammation and fibrogenesis while promoting re-epithelialization[1].

Molecular Weight

441.35

Formula

C23H22Cl2N4O
CAS No.
Appearance

Solid

Color

White to off-white

SMILES

O=C(C1=NN(C2=C(C=C(Cl)C=C2)Cl)C3=C1CC4=CC(C)=CC=C34)NN5CCCCC5
Shipping

Room temperature in continental US; may vary elsewhere.
Storage

4°C, protect from light

*In solvent : -80°C, 6 months; -20°C, 1 month (protect from light)

Solvent & Solubility
In Vitro: 

DMSO : 125 mg/mL (283.22 mM; Need ultrasonic; Hygroscopic DMSO has a significant impact on the solubility of product, please use newly opened DMSO)

Preparing
Stock Solutions
Concentration Solvent Mass 1 mg 5 mg 10 mg
1 mM 2.2658 mL 11.3289 mL 22.6578 mL
5 mM 0.4532 mL 2.2658 mL 4.5316 mL
View the Complete Stock Solution Preparation Table

* Please refer to the solubility information to select the appropriate solvent. Once prepared, please aliquot and store the solution to prevent product inactivation from repeated freeze-thaw cycles.
Storage method and period of stock solution: -80°C, 6 months; -20°C, 1 month (protect from light). When stored at -80°C, please use it within 6 months. When stored at -20°C, please use it within 1 month.

  • Molarity Calculator

  • Dilution Calculator

Mass (g) = Concentration (mol/L) × Volume (L) × Molecular Weight (g/mol)

Mass
=
Concentration
×
Volume
×
Molecular Weight *

Concentration (start) × Volume (start) = Concentration (final) × Volume (final)

This equation is commonly abbreviated as: C1V1 = C2V2

Concentration (start)

C1

×
Volume (start)

V1

=
Concentration (final)

C2

×
Volume (final)

V2

In Vivo Dissolution Calculator
Please enter the basic information of animal experiments:

Dosage

mg/kg

Animal weight
(per animal)

g

Dosing volume
(per animal)

μL

Number of animals

Recommended: Prepare an additional quantity of animals to account for potential losses during experiments.
Calculation results:
Working solution concentration: mg/mL
Purity & Documentation
References

Complete Stock Solution Preparation Table

* Please refer to the solubility information to select the appropriate solvent. Once prepared, please aliquot and store the solution to prevent product inactivation from repeated freeze-thaw cycles.
Storage method and period of stock solution: -80°C, 6 months; -20°C, 1 month (protect from light). When stored at -80°C, please use it within 6 months. When stored at -20°C, please use it within 1 month.

Optional Solvent Concentration Solvent Mass 1 mg 5 mg 10 mg 25 mg
DMSO 1 mM 2.2658 mL 11.3289 mL 22.6578 mL 56.6444 mL
5 mM 0.4532 mL 2.2658 mL 4.5316 mL 11.3289 mL
10 mM 0.2266 mL 1.1329 mL 2.2658 mL 5.6644 mL
15 mM 0.1511 mL 0.7553 mL 1.5105 mL 3.7763 mL
20 mM 0.1133 mL 0.5664 mL 1.1329 mL 2.8322 mL
25 mM 0.0906 mL 0.4532 mL 0.9063 mL 2.2658 mL
30 mM 0.0755 mL 0.3776 mL 0.7553 mL 1.8881 mL
40 mM 0.0566 mL 0.2832 mL 0.5664 mL 1.4161 mL
50 mM 0.0453 mL 0.2266 mL 0.4532 mL 1.1329 mL
60 mM 0.0378 mL 0.1888 mL 0.3776 mL 0.9441 mL
80 mM 0.0283 mL 0.1416 mL 0.2832 mL 0.7081 mL
100 mM 0.0227 mL 0.1133 mL 0.2266 mL 0.5664 mL
  • No file chosen (Maximum size is: 1024 Kb)
  • If you have published this work, please enter the PubMed ID.
  • Your name will appear on the site.

GP1a Related Classifications

Help & FAQs
  • Do most proteins show cross-species activity?

    Species cross-reactivity must be investigated individually for each product. Many human cytokines will produce a nice response in mouse cell lines, and many mouse proteins will show activity on human cells. Other proteins may have a lower specific activity when used in the opposite species.

Keywords:

GP1a511532-96-0Cannabinoid Receptorcannabinoid receptor 2CB2skin wound healinginflammationfibrogenesisre-epithelializationInhibitorinhibitorinhibit

Your Recently Viewed Products:

Inquiry Online

Your information is safe with us. * Required Fields.

Product Name

  

Salutation

Applicant Name *

 

Email Address *

Phone Number *

 

Organization Name *

Department *

 

Requested quantity *

Country or Region *

      

Remarks

Bulk Inquiry

Inquiry Information

Product Name:
GP1a
Cat. No.:
HY-110050
Quantity:
MCE Japan Authorized Agent:

Customer Review

Thank You for Your Feedback!

Request for HNMR Report

Please fill out this form to request the QC report. We will send it to your Email address shortly.

Your information is safe with us. * Required Fields.

Product Name

  

Lot #

Applicant Name *

 

Email Address *

Phone Number

 

Department *

Organization Name *

 

Country or Region *

Remarks

Request for HNMR Report

We have received your request and will respond to you as soon as possible.