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GpTx-1

GpTx-1 is a peptide-based NaV1.7 sodium channel antagonist isolated from the venom of the Chilean spider Grammostola porter. GpTx-1 demonstrates potent inhibitory activity against the NaV1.7 channel with an IC50 value of 10 nM, while exhibiting excellent selectivity for NaV1.4 (IC50 = 0.301 μM) and NaV1.5 (IC50 = 4.20 μM), showing >20-fold and >950-fold selectivity respectively.

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  • CAS No.: 1661050-12-9
  • Formula: C176H271N53O45S7
  • Molecular Weight:4073.82
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    Please store the product under the recommended conditions in the Certificate of Analysis.

  • GpTx-1 Chemical Structure
    GpTx-1 Chemical Structure
CAS No.: 1661050-12-9
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609-228-6898
[email protected] [email protected]
Find Your Local Distributor Your local distributor: Hycultec GmbHHycultec
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All Sodium Channel Isoforms

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  • GpTx-1 Chemical Structure
    GpTx-1 Chemical Structure
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  • GpTx-1