2. GPCR/G Protein Neuronal Signaling
  3. Opioid Receptor
  4. GSK1521498 free base (hydrochloride)

GSK1521498 free base (hydrochloride) is a potent and selective μ-opioid receptor (MOR) antagonist. GSK1521498 free base (hydrochloride) is being used for the treatment of disorders of compulsive consumption of food, alcohol, and agents.

For research use only. We do not sell to patients.

GSK1521498 free base (hydrochloride) Chemical Structure

GSK1521498 free base (hydrochloride) Chemical Structure

CAS No. : 1007578-24-6

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GSK1521498 free base (hydrochloride) Related Antibodies

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Description

GSK1521498 free base (hydrochloride) is a potent and selective μ-opioid receptor (MOR) antagonist. GSK1521498 free base (hydrochloride) is being used for the treatment of disorders of compulsive consumption of food, alcohol, and agents[1].

IC50 & Target

μ Opioid Receptor/MOR

 

Molecular Weight

438.90

Formula

C24H21ClF2N4
CAS No.
SMILES

FC1=C(CNC2CC3=C(C=CC=C3)C2)C(F)=CC(C4=CC=CC(C5=NC=NN5)=C4)=C1.[H]Cl
Shipping

Room temperature in continental US; may vary elsewhere.
Storage

Please store the product under the recommended conditions in the Certificate of Analysis.
Purity & Documentation
References
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GSK1521498 free base (hydrochloride) Related Classifications

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The dilution calculator equation

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This equation is commonly abbreviated as: C1V1 = C2V2

Concentration (start) × Volume (start) = Concentration (final) × Volume (final)
× = ×
C1   V1   C2   V2
Help & FAQs
  • Do most proteins show cross-species activity?

    Species cross-reactivity must be investigated individually for each product. Many human cytokines will produce a nice response in mouse cell lines, and many mouse proteins will show activity on human cells. Other proteins may have a lower specific activity when used in the opposite species.

Keywords:

GSK1521498 free base (hydrochloride)1007578-24-6Opioid ReceptorInhibitorinhibitorinhibit

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GSK1521498 free base (hydrochloride)
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