1. Metabolic Enzyme/Protease
  2. Isocitrate Dehydrogenase (IDH)
  3. IDH1 Inhibitor 3

IDH1 Inhibitor 3 

Cat. No.: HY-107977
Handling Instructions

IDH1 Inhibitor 3 (compound 6f) is a mutant isocitric dehydrogenase 1 (IDH1) inhibitor, with an IC50 of 45 nM for IDH1R132H.

For research use only. We do not sell to patients.

IDH1 Inhibitor 3 Chemical Structure

IDH1 Inhibitor 3 Chemical Structure

CAS No. : 2171081-24-4

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Description

IDH1 Inhibitor 3 (compound 6f) is a mutant isocitric dehydrogenase 1 (IDH1) inhibitor, with an IC50 of 45 nM for IDH1R132H[1].

IC50 & Target

IC50: 45 nM (IDH1R132H)[1].

Storage

Please store the product under the recommended conditions in the Certificate of Analysis.

References
Molecular Weight

591.56

Formula

C₃₁H₂₅F₄N₅O₃

CAS No.

2171081-24-4

SMILES

O=C([[email protected]@H](CC1)N(C2=NC=CC(C#N)=C2)C1=O)N([[email protected]@]3(C(NC4CC(F)(F)C4)=O)CCC5=C3C=CC=C5)C6=CC(F)=CC(F)=C6

Shipping

Room temperature in continental US; may vary elsewhere

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The dilution calculator equation

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This equation is commonly abbreviated as: C1V1 = C2V2

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× = ×
C1   V1   C2   V2

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Product Name:
IDH1 Inhibitor 3
Cat. No.:
HY-107977
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IDH1 Inhibitor 3

Cat. No.: HY-107977