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United States

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製品番号: HY-168144

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DJ-53

DJ-53 (compund 68) is an orally active phenylquinoline-based soluble epoxide hydrolase inhibitor.

商品は「研究用試薬」です。人や動物の医療用・臨床診断用・食品用の製品ではありません。
研究用途以外に使用した場合、当社は一切の責任を負いかねます。

分子式: C₂₆H₂₂F₃N₃O₄
分子量:497.47

保管条件:

Please store the product under the recommended conditions in the Certificate of Analysis.

Data Sheet (264 KB)

DJ-53 構造式

価格（税別）

Amount: USD 0.00

* アイテムを追加する前、数量をご選択ください

Use of MCE Products

Strong Fluorescence Signal / Multi-Disciplinary Applications / High Fluorescence Specificity

生物活性
- 製品説明
- IC₅₀ & Target
- Cellular Effect
化学情報
純度とドキュメンテーション
参考文献
Calculators
Help & FAQs
関連分類
Bioz

生物活性

製品説明

DJ-53 (compund 68) is an orally active phenylquinoline-based soluble epoxide hydrolase inhibitor^[1].

IC₅₀ & Target

Epoxide Hydrolase^[1]

Cellular Effect

Cell Line	Type	Value	Description	References
HEK-293T	IC₅₀	>200 μM Compound: 68; DJ-53	Cytotoxicity against HEK293T cells incubated for 48 hrs by CCK8 assay Cytotoxicity against HEK293T cells incubated for 48 hrs by CCK8 assay	[PMID: 39361006]
HepG2	IC₅₀	>200 μM Compound: 68; DJ-53	Cytotoxicity against human HepG2 cells incubated for 48 hrs by CCK8 assay Cytotoxicity against human HepG2 cells incubated for 48 hrs by CCK8 assay	[PMID: 39361006]

化学情報

分子量 497.47
分子式 C₂₆H₂₂F₃N₃O₄
SMILES

COC1=CC(C2=CC3=CC=C(C=C3N=C2)NC(NCC4=CC=C(C=C4)OC(F)(F)F)=O)=CC(OC)=C1
輸送条件

Room temperature in continental US; may vary elsewhere.
保管条件

Please store the product under the recommended conditions in the Certificate of Analysis.

純度とドキュメンテーション

バッチを選択:

純度: 99.98%

Assay: 99.98%

ee.: 99.98%

データシート (264 KB)
COA (2659 KB)
元素分析報告書 (2659 KB)
HNMR (2659 KB)
CNMR (2659 KB)
RP-HPLC (2659 KB)
NP-HPLC (2659 KB)
MS (2659 KB)
LCMS (2659 KB)
IR (2659 KB)
GC (2659 KB)
OR (2659 KB)
SDS-PAGE (2659 KB)
SEC-HPLC (2659 KB)
Other Report (2659 KB)
取扱説明書 (2659 KB)

参考文献

[1]. Ding J, et al. Discovery of Orally Active Phenylquinoline-Based Soluble Epoxide Hydrolase Inhibitors with Anti-Inflammatory and Analgesic Activity. J Med Chem. 2024 Oct 24;67(20):18412-18447. [Content Brief]

Calculators

モル濃度計算機

Mass (g) = Concentration (mol/L) × Volume (L) × Molecular Weight (g/mol)

Mass Mass

濃度濃度

体積体積

分子量分子量

希釈計算機

濃度 _(開始) × 体積 _(開始) = 濃度 _(終了) × 体積 _(終了)

濃度 _(開始) 濃度 _(開始)

体積 _(開始) 体積 _(開始)

濃度 _(終了) 濃度 _(終了)

体積 _(終了) 体積 _(終了)

Help & FAQs

How should lyophilized recombinant proteins be reconstituted and stored?

1. Before opening the cap, centrifuge the vial at 13000 rpm for 20-30 seconds. This step will ensure that any lyophilized powder that may have adhered to the cap or walls is collected at the bottom of the vial, minimizing the risk of product loss.

Bioz

Keywords

MOQ

Minimum order quantity

100 mg

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